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121348 98 9 U47700 Research Chemical Intermediates Purity 99% Strongest Effect

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121348 98 9 U47700 Research Chemical Intermediates Purity 99% Strongest Effect

China 121348 98 9 U47700 Research Chemical Intermediates Purity 99% Strongest Effect supplier

Large Image :  121348 98 9 U47700 Research Chemical Intermediates Purity 99% Strongest Effect

Product Details:

Place of Origin: China
Brand Name: DJ
Certification: SGS
Model Number: 01

Payment & Shipping Terms:

Minimum Order Quantity: 1g
Price: Negotiation
Packaging Details: 1kg/Aluminum foil bag
Delivery Time: 1-3 work days
Payment Terms: T/T, Western Union, MoneyGram, Bitcion
Supply Ability: 500 Kilogram/Month
Detailed Product Description
Purity: 99% Appearance: White Powder
Colour: White Cas Number: 121348-98-9
Application: Research Chemical Storage: Store In A Cool Dry Place
Formula: C16H22Cl2N2O

U-47700 is an opioid analgesic drug developed by a team at Upjohn in the 1970s that acts as a selective agonist of the µ-opioid receptor with a Kd value of 5.3 nM compared to 910 nM for the κ-opioid receptor and has around 7.5 x the potency of morphine in animal models.

 

U-47700 is a structural isomer of the earlier opioid AH-7921 and the result of a great deal of work elucidating the quantitative structure–activity relationship of the scaffold.

 

Upjohn looked for the key moieties which gave the greatest activity[8] and posted over a dozen patents on related compounds, each optimizing one moiety] until they discovered that U-47700 was the most active.

 

U-47700 became the lead compound of selective kappa-opioid receptor ligands such as U-50488, U-51754 (containing a single methylene spacer difference) and U-69,593, which share very similar structures. Although not used medically, the selective kappa ligands are used in research.

 

121348 98 9 U47700 Research Chemical Intermediates Purity 99% Strongest Effect

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